Our Triptorelin 2mg is freeze-dried Triptorelin in a 2mg vial. Triptorelin is a GnRH (gonadotropin releasing hormone) agonist. It’s for lab research use only.
About Triptorelin
Triptorelin is a ten-amino-acid analog of GnRH, the hypothalamic hormone that drives the pituitary to release LH and FSH. Swapping the glycine at position 6 for D-tryptophan makes it far more potent and longer-lasting than natural GnRH.
It’s an approved drug in long-acting forms for prostate cancer, endometriosis and early puberty, sold as Trelstar and Decapeptyl. In the lab it’s a standard way to switch the reproductive axis on or off.
Buy Triptorelin 2mg online with free shipping
Raw Amino keeps Triptorelin 2mg in stock at $34. When you order, you get:
- Free shipping on every order, to any country we deliver to
- First order? Use code firstrawamino$$ for 10% off
- Pay with crypto and get 15% off at checkout
- Currently in stock; every vial ships sealed and labelled
Triptorelin mechanism of action
A single dose of triptorelin acts like a strong GnRH pulse. The pituitary dumps LH and FSH, which then drive testosterone or estrogen production. Researchers call this the flare effect.
Continuous exposure does the opposite. The GnRH receptors are pulled inside the cell and the pituitary stops responding, so LH, FSH and sex hormones drop. That’s how the long-acting drug forms work.
Triptorelin 2mg at a glance
- Compound: Triptorelin
- Also known as: GnRH agonist, D-Trp6-LHRH
- CAS number: 57773-63-4
- Molecular formula: C64H82N18O13
- Molar mass: 1,311.5 g/mol
- Sequence: pGlu-His-Trp-Ser-Tyr-D-Trp-Leu-Arg-Pro-Gly-NH2
- Amount: 2mg per vial
- Form: freeze-dried (lyophilized) powder in a sealed glass vial
- SKU: RA-TRIPTORELIN-2MG
- Stock: in stock
- Use: laboratory research only
Triptorelin research
Clinical studies over decades cover prostate cancer, endometriosis and central precocious puberty. Single short-acting doses are also used in fertility work to trigger final egg maturation.
In research, labs use it to study how the pituitary responds to GnRH and how that response shuts down with continuous exposure.
For abstracts and full papers, use this PubMed search run by the National Library of Medicine.
Alternatives to Triptorelin
Triptorelin is a long-acting GnRH agonist that first stimulates, then shuts down, LH and FSH. The compounds it’s usually compared with:
- TRH is the three-amino-acid hormone that tells the pituitary to release TSH
- Kisspeptin-10 sits at the top of the reproductive axis and triggers GnRH release
- Oxytocin is the nine-amino-acid hormone behind labor, milk release and social bonding
- Gonadorelin is natural-sequence GnRH, short-lived and pulse-like
- PT-141 is a melanocortin agonist derived from Melanotan II, acting on MC4 receptors in the brain
Each one works on its own hormone pathway, so they aren’t interchangeable. See them side by side on our hormone peptides page.
Triptorelin 2mg mixing chart
Work out concentration by dividing what’s in the vial by the water you add. For example:
- 2mg vial plus 1mL of water: 2mg per mL
- 2mg vial plus 2mL of water: 1mg per mL
Use sterile bacteriostatic water and add it slowly against the glass, not straight onto the powder. Swirl or roll the vial until nothing is left at the bottom. Give it a minute or two if it’s slow; never shake it.
Mark the vial with what you added and when, so nobody has to guess later.
How to keep Triptorelin 2mg stable
Put unopened Triptorelin 2mg in the freezer at -20°C and keep it in its box. The dry powder handles a few days at room temperature in the post without trouble.
After reconstitution it belongs in the fridge (2 to 8°C), and most labs finish it within 28 days. Only mix one vial at a time; powder lasts far longer than solution.
The Triptorelin 2mg label
Each vial carries the Raw Amino logo, the compound name and a purple Research use only band, with the amount (2mg) shown on the label. Check those details when the box arrives and keep the vial sealed until you need it.
The powder inside should look like a small dry cake or loose white flakes at the bottom of the glass. It’s normal for it to shift around in transit or to sit as a thin film on the side of the vial.
If your protocol requires in-house confirmation, set a little material aside from the first vial for your own analysis before the study starts.
Related hormone peptides
- Testagen 20mg: a bioregulator peptide
- Thyrotropin TRH 25mg (Protirelin): a thyrotropin-releasing hormone (TRH)
- PT-141 (Bremelanotide) 10mg: a melanocortin agonist
- Gonadorelin (GnRH) 10mg: a synthetic GnRH
- Oxytocin 10mg: a neuropeptide hormone
Browse all hormone peptides, or open the full Raw Amino shop to see every vial we sell.
Triptorelin 2mg questions and answers
How much is in the Triptorelin 2mg vial?
2mg of freeze-dried Triptorelin. The amount is printed on the label.
Is Triptorelin 2mg in stock?
Yes. It’s in stock now.
Do you ship internationally?
Yes. Raw Amino ships to customers around the world at no charge.
Is there a discount code?
Yes. New customers can use firstrawamino$$ for 10% off, and crypto payments get 15% off at checkout.
What do I mix Triptorelin 2mg with?
Sterile bacteriostatic water. The mixing chart above shows the concentration you get from each volume.
Get Triptorelin 2mg with free shipping
Order Triptorelin 2mg now for $34. Delivery is free, and paying with crypto takes another 15% off.
Need more for the same project? Look through the hormone peptides.
Raw Amino sells this product for laboratory research only. It isn’t for human or veterinary use, and these statements haven’t been evaluated by the FDA.





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